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Cinolazepam

Shí Wikipedia, njikotá édémédé nke onyobulạ
<span title="International nonproprietary name (INN): <nowiki>Cinolazepam</nowiki>">Cinolazepam
Clinical data
Trade names Gerodorm
AHFS/Drugs.com cinolazepam
Routes of



administration
Oral
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  • N05CD13 (WHO)
Ọnọdụ iwu
Ọnọdụ iwu
  • US: Enweghị usoro
Ihe omuma pharmacokinetic
Bioavailability 90-100%
Metabolism Ọrịa imeju
<span class="nowrap">Ọkara ndụ</span> e wepụrụ awa 3.8[1]
Mgbapụta Akụrụ
Ihe ndị na-eme ka a mata ya
Aha IUPAC
  • (RS) -3-[9-Chloro-6- (2-fluorophenyl) -4-hydroxy-3-oxo-2,5-diazabicyclo[5.4.0]undeca-5,8,10,12-tetraen-2-yl]prenitopanrile
Nọmba CAS
PubChem <abbr title="<nowiki>Compound ID</nowiki>">CID
Ụlọ Akụ̀ Ọgwụ
ChemSpider
UNII
KEGG
ChEBI
  • CHEBI:59514 Ycheck
ChEMBL
Ihe omuma kemịkal na nke anụ ahụ
Nhazi C18H13ClFN3O2
Ọkpụkpụ nke ọkpụkpụ 357.8 g·mol-1
Ihe nlereanya 3D (JSmol)
Chirality Ngwakọta agbụrụ
Mmetụta ihere
  • FC1=CC=C1C2=NC (C (N (CCC#N) C3=C2C=C (C=C3) Cl) =O) O
InChI
  • InChI=1S/C18H13ClFN3O2/c19-11-6-7-15-13 (10-11) 16 (12-4-1-2-5-14 (12) 20) 22-17 (24) 18 (25) 23 (15) 9-3-8-21/h1-2,4-7,10,17,24H,3,9H2 Ycheck
  • Isi:XAXMYcheckHMKTCNRRZ-UHFFFAOYSA-N Y
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Cinolazepam[2] (nke a na-ere n'okpuru aha Gerodorm) bụ ọgwụ nke bụ benzodiazepine.[3] Ọ nwere ihe na-eme ka nchegbu kwụsị, ihe na-egbochi nkụchi, ihe na'ime ka ọ dị jụụ na ihe na-ehi ụra. N'ihi ikike ya ahazi na ụdị nke ụwa na ụdị ke amụta site na iji Tinye na Enyi siri ike, a na-eji ya eme ihe dị ka ọgwụ na-eme ka mmadụ kwụsị.

E nyere ya ikike n'afọ 1978 ma malite iji ya mee ihe n'ụzọ ọgwụ na 1992.[4] A kwadoghị Cinolazepam maka ire ere na United States ma ọ bụ Canada.

Ntụaka

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  1. "ZUSAMMENFASSUNG DER MERKMALE DES ARZNEIMITTELS" (Press release). (in Austrian German). Austria: G.L. Pharma GmbH. Bundesamt für Sicherheit im Gesundheitswesen. October 2018. Archived from the original on 2019-01-02. Retrieved 2019-01-02.
  2. US Patent 4388313 Novel 3-hydroxy-1,4-benzodiazepine-2-ones and process for the preparation thereof
  3. Lannacher Romania (1999). Gerodorm (ro). Produse Gerot inregistrate in Romania. Archived from the original on 11 October 2006. Retrieved on 17 August 2006.
  4. (2006) Analogue-based Drug Discovery (in en). John Wiley & Sons. ISBN 9783527607495. 

Njikọ mpụga

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Templeeti:BenzodiazepinesTempleeti:GABAAR PAMs